食品研究与开发
食品研究與開髮
식품연구여개발
FOOD RESEARCH AND CEVELOPMENT
2013年
11期
97-100
,共4页
玄红专%李振%付崇罗%桑青
玄紅專%李振%付崇囉%桑青
현홍전%리진%부숭라%상청
咖啡酸苯乙酯(CAPE)%蜂胶%抗肿瘤%分子机制
咖啡痠苯乙酯(CAPE)%蜂膠%抗腫瘤%分子機製
가배산분을지(CAPE)%봉효%항종류%분자궤제
caffeic acid phenethyl ester%propolis%antitumor%molecular mechanism
咖啡酸苯乙酯(CAPE)是蜂胶中的一种活性组分,长期在民间医药中使用,具有多种生物学活性。CAPE抑制肿瘤细胞生长是近年来的研究热点。本文主要综述CAPE对多种肿瘤的抑制功效及其抗肿瘤的分子机制,指出CAPE主要通过清除ROS,抑制NF-κB,诱导细胞周期阻滞及诱导肿瘤细胞凋亡来抑制肿瘤的生长。表明CAPE作为一种潜在的抗肿瘤药物具有广阔的应用前景。
咖啡痠苯乙酯(CAPE)是蜂膠中的一種活性組分,長期在民間醫藥中使用,具有多種生物學活性。CAPE抑製腫瘤細胞生長是近年來的研究熱點。本文主要綜述CAPE對多種腫瘤的抑製功效及其抗腫瘤的分子機製,指齣CAPE主要通過清除ROS,抑製NF-κB,誘導細胞週期阻滯及誘導腫瘤細胞凋亡來抑製腫瘤的生長。錶明CAPE作為一種潛在的抗腫瘤藥物具有廣闊的應用前景。
가배산분을지(CAPE)시봉효중적일충활성조분,장기재민간의약중사용,구유다충생물학활성。CAPE억제종류세포생장시근년래적연구열점。본문주요종술CAPE대다충종류적억제공효급기항종류적분자궤제,지출CAPE주요통과청제ROS,억제NF-κB,유도세포주기조체급유도종류세포조망래억제종류적생장。표명CAPE작위일충잠재적항종류약물구유엄활적응용전경。
@@@@Caffeic acid phenethyl ester (CAPE) is a biologically active component of propolis from honeybee hives. It has been used in folk medicine since ancient time ,and has widely biological propertities. CAPE can suppress reproductive of many kinds of tumors,and has been a hot topic in recent years. The antitumor activities of CAPE and its molecular mechanisms were reviewed in this article ,the results indicated that CAPE suppressed tumor reproductive by ROS scavenging,pro-oxidative activity,NF-κB inhibition,cell cycle inhibition and apoptosis induction. It can be conclude that CAPE has widely application as a potential antitumor drug.